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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4246 | Varenicline dihydrochloride | AChR | |
Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist. | |||
T5678 | Lazabemide hydrochloride | N-(2-Aminoethyl)-5-chlor-2-pyridincarbox | MAO , Monoamine Oxidase |
Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki:7.9nM). | |||
T5470 | LAZABEMIDE | Ro 19-6327 | MAO , Monoamine Oxidase |
Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). | |||
T1657 | Varenicline Tartrate | Champix tartrate,Chantix tartrate,CP 526555-18 | AChR |
Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESSATION. | |||
T22357 | Lobeline sulfate | Lobelin sulphate | Others |
Lobelin sulphate is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in insomnia, and smoking cessation, peripheral va... | |||
T32833 | Lobeline, (+)- | (+)-Lobeline | |
Lobeline, (+)- is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has been proposed for a variety of therapeutic uses including in respiratory disorders, periphe... | |||
T70625 | Nicotine lactate | ||
Nicotine is a naturally produced alkaloid in the nightshade family of plants (most predominantly in tobacco and Duboisia hopwoodii) and is widely used recreationally as a stimulant and anxiolytic. As a pharmaceutical dru... | |||
T80219 | α-Conotoxin TxID | ||
α-Conotoxin TxID is a potent antagonist of the α3β4 nicotinic acetylcholine receptor (nAChR), exhibiting an inhibitory half-maximal inhibitory concentration (IC50) of 12.5 nM. Its inhibitory activity against the closely ... | |||
TC0022 | Desoxypeganine | Deoxypeganine | AChE |
Desoxypeganine (Deoxypeganine) is an inhibitor of cholinesterase. It acting preferentially on butyrylcholinesterase, and as a selective inhibitor of monoamine oxidase A but not monoamine oxidase B.Desoxypeganine is being... | |||
T4246L | Varenicline | ||
Varenicline (CP 526555), a cytisine-based nicotinic ligand, is a potent partial agonist for the α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM and acts as a full agonist for α7 and α3β4 nAChRs... |